LATP
LATP:
Two leading products (LTP-03, and LTP-0401) are in early pre-clinical stage. The efficacy and toxicity were confirmed in rodent studies. IND-enabling studies of LTP-03 has been in progress
LTP-03
- Balanced GLP-1R and GCGR activation, and enhanced GIPR activation
- All naturalamino acid and no chemical modifacations renders low immunogenicity
- MininalCNS exposure, mild effect on food intake
- Half-life similar to Semaglutide in mice; Co-administration with Sitagliptin (a DPPIV inhibitor) further extended the half-life.
- Mimic physiological properties of native peptides: no sustained activation of related receptors
- Similar physiochemical and pharmacological profiles, and CMC to Dulaglutide
- Potentially armed with additional metabolic hormones
LTP-0521
- Reduced GCGR activation with enhanced GIPR activation
- Similar to native sequence and containing only natural amino acids, thus decreasing any immunogenicity risk
- Monovalent analogs mimic physiological properties of native peptides, no sustained activation of related receptors
- Minimal CNS exposure, mild effect on food intake
- Prolonged half-life
- Similar physiochemical and pharmacological profiles, and CMC to Dulaglutide